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---
license: mit
pretty_name: Drug-Likeness RDKit Dataset
tags:
- cheminformatics
- rdkit
- drug-likeness
- AutoML
configs:
- config_name: default
  data_files:
  - split: train_rdkit
    path: data/train_rdkit-*
  - split: test_rdkit
    path: data/test_rdkit-*
dataset_info:
  features:
  - name: label
    dtype: int64
  - name: Standardized_SMILES
    dtype: string
  - name: MaxAbsEStateIndex
    dtype: float64
  - name: MaxEStateIndex
    dtype: float64
  - name: MinAbsEStateIndex
    dtype: float64
  - name: MinEStateIndex
    dtype: float64
  - name: qed
    dtype: float64
  - name: SPS
    dtype: float64
  - name: MolWt
    dtype: float64
  - name: HeavyAtomMolWt
    dtype: float64
  - name: ExactMolWt
    dtype: float64
  - name: NumValenceElectrons
    dtype: int64
  - name: NumRadicalElectrons
    dtype: int64
  - name: MaxPartialCharge
    dtype: float64
  - name: MinPartialCharge
    dtype: float64
  - name: MaxAbsPartialCharge
    dtype: float64
  - name: MinAbsPartialCharge
    dtype: float64
  - name: FpDensityMorgan1
    dtype: float64
  - name: FpDensityMorgan2
    dtype: float64
  - name: FpDensityMorgan3
    dtype: float64
  - name: BCUT2D_MWHI
    dtype: float64
  - name: BCUT2D_MWLOW
    dtype: float64
  - name: BCUT2D_CHGHI
    dtype: float64
  - name: BCUT2D_CHGLO
    dtype: float64
  - name: BCUT2D_LOGPHI
    dtype: float64
  - name: BCUT2D_LOGPLOW
    dtype: float64
  - name: BCUT2D_MRHI
    dtype: float64
  - name: BCUT2D_MRLOW
    dtype: float64
  - name: AvgIpc
    dtype: float64
  - name: BalabanJ
    dtype: float64
  - name: BertzCT
    dtype: float64
  - name: Chi0
    dtype: float64
  - name: Chi0n
    dtype: float64
  - name: Chi0v
    dtype: float64
  - name: Chi1
    dtype: float64
  - name: Chi1n
    dtype: float64
  - name: Chi1v
    dtype: float64
  - name: Chi2n
    dtype: float64
  - name: Chi2v
    dtype: float64
  - name: Chi3n
    dtype: float64
  - name: Chi3v
    dtype: float64
  - name: Chi4n
    dtype: float64
  - name: Chi4v
    dtype: float64
  - name: HallKierAlpha
    dtype: float64
  - name: Ipc
    dtype: float64
  - name: Kappa1
    dtype: float64
  - name: Kappa2
    dtype: float64
  - name: Kappa3
    dtype: float64
  - name: LabuteASA
    dtype: float64
  - name: PEOE_VSA1
    dtype: float64
  - name: PEOE_VSA10
    dtype: float64
  - name: PEOE_VSA11
    dtype: float64
  - name: PEOE_VSA12
    dtype: float64
  - name: PEOE_VSA13
    dtype: float64
  - name: PEOE_VSA14
    dtype: float64
  - name: PEOE_VSA2
    dtype: float64
  - name: PEOE_VSA3
    dtype: float64
  - name: PEOE_VSA4
    dtype: float64
  - name: PEOE_VSA5
    dtype: float64
  - name: PEOE_VSA6
    dtype: float64
  - name: PEOE_VSA7
    dtype: float64
  - name: PEOE_VSA8
    dtype: float64
  - name: PEOE_VSA9
    dtype: float64
  - name: SMR_VSA1
    dtype: float64
  - name: SMR_VSA10
    dtype: float64
  - name: SMR_VSA2
    dtype: float64
  - name: SMR_VSA3
    dtype: float64
  - name: SMR_VSA4
    dtype: float64
  - name: SMR_VSA5
    dtype: float64
  - name: SMR_VSA6
    dtype: float64
  - name: SMR_VSA7
    dtype: float64
  - name: SMR_VSA8
    dtype: float64
  - name: SMR_VSA9
    dtype: float64
  - name: SlogP_VSA1
    dtype: float64
  - name: SlogP_VSA10
    dtype: float64
  - name: SlogP_VSA11
    dtype: float64
  - name: SlogP_VSA12
    dtype: float64
  - name: SlogP_VSA2
    dtype: float64
  - name: SlogP_VSA3
    dtype: float64
  - name: SlogP_VSA4
    dtype: float64
  - name: SlogP_VSA5
    dtype: float64
  - name: SlogP_VSA6
    dtype: float64
  - name: SlogP_VSA7
    dtype: float64
  - name: SlogP_VSA8
    dtype: float64
  - name: SlogP_VSA9
    dtype: float64
  - name: TPSA
    dtype: float64
  - name: EState_VSA1
    dtype: float64
  - name: EState_VSA10
    dtype: float64
  - name: EState_VSA11
    dtype: float64
  - name: EState_VSA2
    dtype: float64
  - name: EState_VSA3
    dtype: float64
  - name: EState_VSA4
    dtype: float64
  - name: EState_VSA5
    dtype: float64
  - name: EState_VSA6
    dtype: float64
  - name: EState_VSA7
    dtype: float64
  - name: EState_VSA8
    dtype: float64
  - name: EState_VSA9
    dtype: float64
  - name: VSA_EState1
    dtype: float64
  - name: VSA_EState10
    dtype: float64
  - name: VSA_EState2
    dtype: float64
  - name: VSA_EState3
    dtype: float64
  - name: VSA_EState4
    dtype: float64
  - name: VSA_EState5
    dtype: float64
  - name: VSA_EState6
    dtype: float64
  - name: VSA_EState7
    dtype: float64
  - name: VSA_EState8
    dtype: float64
  - name: VSA_EState9
    dtype: float64
  - name: FractionCSP3
    dtype: float64
  - name: HeavyAtomCount
    dtype: int64
  - name: NHOHCount
    dtype: int64
  - name: NOCount
    dtype: int64
  - name: NumAliphaticCarbocycles
    dtype: int64
  - name: NumAliphaticHeterocycles
    dtype: int64
  - name: NumAliphaticRings
    dtype: int64
  - name: NumAmideBonds
    dtype: int64
  - name: NumAromaticCarbocycles
    dtype: int64
  - name: NumAromaticHeterocycles
    dtype: int64
  - name: NumAromaticRings
    dtype: int64
  - name: NumAtomStereoCenters
    dtype: int64
  - name: NumBridgeheadAtoms
    dtype: int64
  - name: NumHAcceptors
    dtype: int64
  - name: NumHDonors
    dtype: int64
  - name: NumHeteroatoms
    dtype: int64
  - name: NumHeterocycles
    dtype: int64
  - name: NumRotatableBonds
    dtype: int64
  - name: NumSaturatedCarbocycles
    dtype: int64
  - name: NumSaturatedHeterocycles
    dtype: int64
  - name: NumSaturatedRings
    dtype: int64
  - name: NumSpiroAtoms
    dtype: int64
  - name: NumUnspecifiedAtomStereoCenters
    dtype: int64
  - name: Phi
    dtype: float64
  - name: RingCount
    dtype: int64
  - name: MolLogP
    dtype: float64
  - name: MolMR
    dtype: float64
  - name: fr_Al_COO
    dtype: int64
  - name: fr_Al_OH
    dtype: int64
  - name: fr_Al_OH_noTert
    dtype: int64
  - name: fr_ArN
    dtype: int64
  - name: fr_Ar_COO
    dtype: int64
  - name: fr_Ar_N
    dtype: int64
  - name: fr_Ar_NH
    dtype: int64
  - name: fr_Ar_OH
    dtype: int64
  - name: fr_COO
    dtype: int64
  - name: fr_COO2
    dtype: int64
  - name: fr_C_O
    dtype: int64
  - name: fr_C_O_noCOO
    dtype: int64
  - name: fr_C_S
    dtype: int64
  - name: fr_HOCCN
    dtype: int64
  - name: fr_Imine
    dtype: int64
  - name: fr_NH0
    dtype: int64
  - name: fr_NH1
    dtype: int64
  - name: fr_NH2
    dtype: int64
  - name: fr_N_O
    dtype: int64
  - name: fr_Ndealkylation1
    dtype: int64
  - name: fr_Ndealkylation2
    dtype: int64
  - name: fr_Nhpyrrole
    dtype: int64
  - name: fr_SH
    dtype: int64
  - name: fr_aldehyde
    dtype: int64
  - name: fr_alkyl_carbamate
    dtype: int64
  - name: fr_alkyl_halide
    dtype: int64
  - name: fr_allylic_oxid
    dtype: int64
  - name: fr_amide
    dtype: int64
  - name: fr_amidine
    dtype: int64
  - name: fr_aniline
    dtype: int64
  - name: fr_aryl_methyl
    dtype: int64
  - name: fr_azide
    dtype: int64
  - name: fr_azo
    dtype: int64
  - name: fr_barbitur
    dtype: int64
  - name: fr_benzene
    dtype: int64
  - name: fr_benzodiazepine
    dtype: int64
  - name: fr_bicyclic
    dtype: int64
  - name: fr_diazo
    dtype: int64
  - name: fr_dihydropyridine
    dtype: int64
  - name: fr_epoxide
    dtype: int64
  - name: fr_ester
    dtype: int64
  - name: fr_ether
    dtype: int64
  - name: fr_furan
    dtype: int64
  - name: fr_guanido
    dtype: int64
  - name: fr_halogen
    dtype: int64
  - name: fr_hdrzine
    dtype: int64
  - name: fr_hdrzone
    dtype: int64
  - name: fr_imidazole
    dtype: int64
  - name: fr_imide
    dtype: int64
  - name: fr_isocyan
    dtype: int64
  - name: fr_isothiocyan
    dtype: int64
  - name: fr_ketone
    dtype: int64
  - name: fr_ketone_Topliss
    dtype: int64
  - name: fr_lactam
    dtype: int64
  - name: fr_lactone
    dtype: int64
  - name: fr_methoxy
    dtype: int64
  - name: fr_morpholine
    dtype: int64
  - name: fr_nitrile
    dtype: int64
  - name: fr_nitro
    dtype: int64
  - name: fr_nitro_arom
    dtype: int64
  - name: fr_nitro_arom_nonortho
    dtype: int64
  - name: fr_nitroso
    dtype: int64
  - name: fr_oxazole
    dtype: int64
  - name: fr_oxime
    dtype: int64
  - name: fr_para_hydroxylation
    dtype: int64
  - name: fr_phenol
    dtype: int64
  - name: fr_phenol_noOrthoHbond
    dtype: int64
  - name: fr_phos_acid
    dtype: int64
  - name: fr_phos_ester
    dtype: int64
  - name: fr_piperdine
    dtype: int64
  - name: fr_piperzine
    dtype: int64
  - name: fr_priamide
    dtype: int64
  - name: fr_prisulfonamd
    dtype: int64
  - name: fr_pyridine
    dtype: int64
  - name: fr_quatN
    dtype: int64
  - name: fr_sulfide
    dtype: int64
  - name: fr_sulfonamd
    dtype: int64
  - name: fr_sulfone
    dtype: int64
  - name: fr_term_acetylene
    dtype: int64
  - name: fr_tetrazole
    dtype: int64
  - name: fr_thiazole
    dtype: int64
  - name: fr_thiocyan
    dtype: int64
  - name: fr_thiophene
    dtype: int64
  - name: fr_unbrch_alkane
    dtype: int64
  - name: fr_urea
    dtype: int64
  splits:
  - name: train_rdkit
    num_bytes: 14788191
    num_examples: 8234
  - name: test_rdkit
    num_bytes: 12413665
    num_examples: 6913
  download_size: 10842785
  dataset_size: 27201856
---

# Drug-Likeness Prediction Dataset (Based on DBPP-Predictor Data)

This dataset was created as part of a final project on drug-likeness prediction, based on the data from the DBPP-Predictor paper:

> Gu, Y., Wang, Y., Zhu, K. et al. DBPP-Predictor: a novel strategy for prediction of chemical drug-likeness based on property profiles. J Cheminform 16, 4 (2024). https://doi.org/10.1186/s13321-024-00800-9

 It includes curated molecular data, preprocessed RDKit descriptors, and training/test splits suitable for training classification models to distinguish drug-like from non-drug-like molecules.

## Project Background

Drug-likeness refers to the potential of a small molecule to become a drug. Traditional rule-based approaches (e.g., Lipinski's Rule of Five) often fail to generalize across complex compounds. This project uses RDKit descriptors and AutoML (H2O) to construct a highly interpretable, generalizable classification model.

## Dataset Description

The dataset is derived from the DBPP GitHub repository (https://github.com/yxgu2353/DBPP-Predictor.git). It includes:
- 5,147 drug-like molecules (FDA and globally approved drugs)
- 10,000 non-drug-like molecules sampled from ZINC

All molecules were standardized using MolVS(clean_data.py), the datasets were split by sklearn(split_dataset.py), and RDKit descriptors (216 features) were computed (Rdkit_descriptor.py).

### Files:
- 'train_rdkit_descriptors.parquet'
- 'test_rdkit_descriptors.parquet'

Each file contains:
- 'label': 0 for non-drug, 1 for drug
- 'Standardized_SMILES'
- 216 numerical RDKit descriptors

## Model Development

All models were trained using H2O AutoML with 10-fold cross-validation(model_constrcution.py). The top 3 models were also evaluated using an independent test set, and SHAP analysis was used to interpret the top structural features contributing to drug-likeness(model_analysis.py).